β-ADRENERGIC BLOCKING AGENTS
1. NONSELECTIVE (β1 and β2)
a. Without intrinsic sympathomimetic
activity
Propranolol
Sotalol
Timolol
b. With intrinsic sympathomimetic
activity
Pindolol
c. With additional α-blocking property
Labetalol
Carvedilol
2. CARDIOSELECTIVE (β1)
Metoprolol
Atenolol
Acebutolol
Bisoprolol
Esmolol
Betaxolol
Celiprolol
Nebivolol
GENERATION WISE CLASSIFICATION
1. First Generation (older, nonselective)
Propranolol
Timolol
Sotalol
Pindolol
2. Second Generation (β2 selective)
Metoprolol
Atenolol
Acebutolol
Bisoprolol
Esmolol
3. Third Generation (with additional α blocking
and/ or vasodilator property)
Labetalol
Carvedilol
Celiprolol
Nabivolol